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Compound | Naringin |
Animal species | rat and human intestinal microflora |
Metabolism parameters | |
Metabolites |
Naringin
|
Crude drug | Citrus Unshiu Peel |
References | 1) Jun-Shik Choi and Keon Wook Kang, Enhanced tamoxifen bioavailability after oral administration of tamoxifen in rats pretreated with naringin. Arch Pharm Res 31: 1631-1636 (2008). DOI 10.1007/s12272-001-2161-7. 2) Xijun Wang, Tetsuro Sakurai, Xi Chen, Hui Sun, Zenghui Wang, Qinglong Sun,Wenjun Sun, Hongxin Cao, Hydrolysis of flavanone glycosides and degradation of the corresponding aglycones from dried immature citrus fruit by human fecal flora in vitro. Planta Med 74: 1751–1755 (2008). |
Remarks | ① tamoxifenの体内動態に及ぼすnaringinの影響をラットを用いて検証した。 ②ヒト腸内細菌フローラによるnaringinの代謝 |